SCHEMBL4655285

SCHEMBL4655285

Cn1ccc2cc(NC(=O)c3cc4ccccc4n3-c3ccc(-c4ccccc4)cc3)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 2/20 0.53
MAOB P27338 1/20 0.46
NOTUM Q6P988 1/20 0.45
TSHR P16473 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HTR2B P41595 3/20 0.45
MEN1 O00255 2/20 0.45
TP53 P04637 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
MAPT P10636 2/20 0.45
CYP2C19 P33261 2/20 0.45
RECQL P46063 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HTR2C P28335 4/20 0.44
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4656220 0.93 ECE1 (0.59) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL4655331 0.89 MAOB (0.51) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL4656319 0.89 ECE1 (0.50) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL4655289 0.88 ECE1 (0.53) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL3571160 0.88 ECE1 (0.48) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL4655301 0.88 ECE1 (0.48) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL4656120 0.87 ECE1 (0.50) ECE1MAOBNOTUMTSHRALDH1A1
SCHEMBL4655241 0.86 NOTUM (0.49) ECE1MAOBNOTUMTSHRHTR2B
SCHEMBL4655315 0.86 ECE1 (0.48) ECE1MAOBNOTUMTSHRHTR2B
SCHEMBL4655291 0.86 ECE1 (0.49) ECE1MAOBNOTUMTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776340-B1 N-(1H-INDOLYL)-H-INDOLE-2-CARB0XAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE SANOFI AVENTIS (FR) 2008-12-03 EP claimed