SCHEMBL4655306

SCHEMBL4655306

O=C(Oc1ccco1)N(Cc1cccc(-c2ccc3ncnc(NC4CC4)c3c2)c1)C1CC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 13/20 0.49
USP2 O75604 4/20 0.48
CYP1A2 P05177 4/20 0.48
CYP3A4 P08684 4/20 0.48
CLK4 Q9HAZ1 4/20 0.48
MAPK1 P28482 3/20 0.48
CYP2C19 P33261 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CYP2D6 P10635 2/20 0.48
ALOX15 P16050 2/20 0.48
LMNA P02545 2/20 0.48
TSHR P16473 1/20 0.48
MAP4K4 O95819 2/20 0.48
PIK3CD O00329 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4171855 0.88 IRAK4 (0.53) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4187738 0.87 CYP1A2 (0.59) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4175372 0.84 IRAK4 (0.55) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4654450 0.84 IRAK4 (0.49) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4173066 0.84 IRAK4 (0.61) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4654418 0.83 CLK4 (0.41) USP2CYP1A2CYP3A4CLK4MAPK1
SCHEMBL13917321 0.83 IRAK4 (0.57) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4177424 0.83 IRAK4 (0.60) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4655430 0.83 IRAK4 (0.48) IRAK4USP2CYP1A2CYP3A4CLK4
SCHEMBL4183839 0.82 IRAK4 (0.59) IRAK4USP2CYP1A2CYP3A4CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996562-A1 SUBSTITUTED 4-AMINO-QUINAZOLINE DERIVATIVES AS REGULATORS OF METABOTROPIC GLUTAMATE RECEPTORS AND THEIR USE FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-12-03 EP disclosed
WO-2007104560-A1 SUBSTITUTED 4-AMINO-QUINAZOLINE DERIVATIVES AS REGULATORS OF METABOTROPIC GLUTAMATE RECEPTORS AND THEIR USE FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-09-20 WO disclosed