SCHEMBL4656304

SCHEMBL4656304

N#CC(C#N)(CCCC(F)(F)F)Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
TAAR1 Q96RJ0 1/20 0.37
IDO1 P14902 3/20 0.36
KIF11 P52732 2/20 0.36
DAO P14920 1/20 0.35
KMT2A Q03164 1/20 0.35
MIF P14174 1/20 0.35
MAOB P27338 3/20 0.34
PYCR1 P32322 1/20 0.33
NAAA Q02083 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657451 0.90 TAAR1 (0.39) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL4657412 0.87 TAAR1 (0.41) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL6840018 0.86 ESR1 (0.37) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL4657501 0.86 ESR1 (0.39) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL4657460 0.86 MAOB (0.36) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL6835187 0.84 ESR1 (0.36) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL4657572 0.84 MAOB (0.36) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL4657483 0.83 TAAR1 (0.43) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL6821464 0.83 ESR1 (0.37) ESR1ESR2TAAR1IDO1KIF11
SCHEMBL6824229 0.82 ESR1 (0.39) ESR1ESR2TAAR1IDO1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 ESR1 4561/4885ESR2 4792/4885TAAR1 644/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 ESR1 4835/4885ESR2 4741/4885TAAR1 632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.