SCHEMBL4659666

SCHEMBL4659666

CC(C)(C)OC(=O)C(c1ccccc1)[C@H](N)CO

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
LTA4H P09960 1/20 0.40
ATM Q13315 2/20 0.39
AAK1 Q2M2I8 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
CYP2D6 P10635 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
RIPK1 Q13546 1/20 0.38
CYP1A2 P05177 1/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KIF11 P52732 1/20 0.38
MAPT P10636 1/20 0.38
SLC7A5 Q01650 1/20 0.37
TNF P01375 1/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3915984 1.00 KMT2A (0.45) KMT2ALTA4HATMAAK1CTSS
SCHEMBL4730837 0.88 KMT2A (0.45) KMT2ALTA4HATMAAK1CTSS
SCHEMBL24851748 0.82 KMT2A (0.52) KMT2AATMAAK1CTSSCTSK
SCHEMBL27598805 0.81 KMT2A (0.47) KMT2ALTA4HATMAAK1CTSS
SCHEMBL6647558 0.81 KMT2A (0.47) KMT2ALTA4HATMAAK1CTSS
SCHEMBL6702668 0.81 KMT2A (0.47) KMT2ALTA4HATMAAK1CTSS
SCHEMBL10952116 0.81 KMT2A (0.39) KMT2ALTA4HATMAAK1CTSS
SCHEMBL6703239 0.80 AAK1 (0.40) KMT2ALTA4HATMAAK1CTSS
SCHEMBL4520911 0.80 KMT2A (0.46) KMT2ALTA4HATMAAK1CTSS
SCHEMBL4526758 0.80 KMT2A (0.46) KMT2ALTA4HATMAAK1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720855-A4 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORP (US) 2008-12-17 EP disclosed
EP-1720855-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-11-15 EP disclosed
WO-2005085227-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2005-09-15 WO disclosed