SCHEMBL4660359

SCHEMBL4660359

CCC(c1cccc(N(C(C)C)C(C)C)c1)c1cc(CO)ccc1OC(=O)c1ccc(OC)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
KMT2A Q03164 5/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
TAS2R14 Q9NYV8 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
TP53 P04637 2/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ACHE P22303 1/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
MEN1 O00255 3/20 0.35
MAPT P10636 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4659036 0.91 CHRM2 (0.51) CHRM2CHRM1KMT2AKEAP1NFE2L2
SCHEMBL4660409 0.91 CHRM2 (0.51) CHRM2CHRM1KMT2AKEAP1NFE2L2
SCHEMBL4660350 0.91 CHRM2 (0.46) CHRM2CHRM1KMT2AESR1ESR2
SCHEMBL4659037 0.90 CHRM2 (0.46) CHRM2CHRM1KMT2ATP53GAA
SCHEMBL4661597 0.88 CHRM2 (0.46) CHRM2CHRM1KMT2AGAAACHE
SCHEMBL4659055 0.86 CHRM2 (0.43) CHRM2CHRM1KMT2AGAATHRB
SCHEMBL4660336 0.85 CHRM2 (0.47) CHRM2CHRM1KMT2AESR1ESR2
SCHEMBL1158251 0.84 CHRM2 (0.62) CHRM2CHRM1KMT2ATP53ACHE
SCHEMBL4659057 0.84 CHRM2 (0.62) CHRM2CHRM1KMT2ATP53ACHE
Hydrochloric Acid SCHEMBL16166361 0.84 CHRM2 (0.61) CHRM2CHRM1KMT2AACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254890-A1 Derivatives of 3,3-diphenylpropylamines SCHWARZ PHARMA AG (DE) 2002-11-06 EP claimed
EP-2004592-A1 SYNTHESIS OF PHENOLIC ESTERS OF HYDROXYMETHYL PHENOLS Schwarz Pharma Ltd. (IE) 2008-12-24 EP disclosed
WO-2007140986-A1 SYNTHESIS OF PHENOLIC ESTERS OF HYDROXYMETHYL PHENOLS SCHWARZ PHARMA LTD (IE) 2007-12-13 WO disclosed