SCHEMBL466114

SCHEMBL466114

Nc1cc(=O)[nH]c(N)n1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1057956 0.76
SCHEMBL7161983 0.76
SCHEMBL8723531 0.76
SCHEMBL908316 0.76
SCHEMBL190318 0.76
Water SCHEMBL8081142 0.75 CYP3A4 (0.59)
Water SCHEMBL9836997 0.75 CYP3A4 (0.59)
SCHEMBL15971206 0.73 CYP3A4 (0.57)
SCHEMBL31231913 0.73 CYP3A4 (0.57)
SCHEMBL3230029 0.73 CYP3A4 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 374 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4547747-A1 POLYOXMETHYLENE POLYMER INCORPORATING AN ALDEHYDE SCAVENGER Colormatrix Holdings, Inc. (US) 2025-05-07 EP claimed
CN-119156419-A Polyoxymethylene polymers containing aldehyde scavengers 彩色矩阵控股公司 2024-12-17 CN claimed
WO-2024003633-A1 POLYOXMETHYLENE POLYMER INCORPORATING AN ALDEHYDE SCAVENGER COLORMATRIX HOLDINGS, INC. (US) 2024-01-04 WO claimed
US-20230312809-A1 LIQUID FORMULATION COMPRISING AN ALDEHYDE SCAVENGER Ferline SA (CH) 2023-10-05 US claimed
EP-4157915-A1 LIQUID FORMULATION COMPRISING AN ALDEHYDE SCAVENGER Ferline SA (CH) 2023-04-05 EP claimed
CN-115698118-A Liquid formulations comprising aldehyde scavengers 佛莱恩股份公司 2023-02-03 CN claimed
WO-2021239634-A1 LIQUID FORMULATION COMPRISING AN ALDEHYDE SCAVENGER REPI S.R.L. (IT) 2021-12-02 WO claimed
US-20160038444-A1 MODULATON OF CELLULAR DNA REPAIR ACTIVITY TO INTERCEPT MALIGNANCY THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-02-11 US claimed
EP-2968371-A2 MODULATION OF CELLULAR DNA REPAIR ACTIVITY TO INTERCEPT MALIGNANCY The Board of Trustees of the Leland Stanford Junior University (US) 2016-01-20 EP claimed
WO-2014164730-A2 MODULATION OF CELLULAR DNA REPAIR ACTIVITY TO INTERCEPT MALIGNANCY THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2014-10-09 WO claimed
EP-1363637-A1 PYRIMIDINE COMPOUNDS AND METHODS FOR MAKING AND USING THE SAME DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 2003-11-26 EP claimed
WO-2003082967-A2 COMPOUNDS USEFUL FOR REDUCING ACETALDEHYDE CONTENT OF POLYETHYLENE TEREPHTHALATE, THEIR USE AND PRODUCTS RESULTING THEREFROM EQUIPOLYMERS GMBH (DE) 2003-10-09 WO claimed
US-20030040524-A1 Pyrimidine compounds and methods for making and using the same GANGJEE ALEEM (US) 2003-02-27 US claimed
WO-2002060450-A1 PYRIMIDINE COMPOUNDS AND METHODS FOR MAKING AND USING THE SAME DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 2002-08-08 WO claimed
EP-1105396-A1 PROCESS FOR THE PREPARATION OF PYRROLO[2,3-D]PYRIMIDINES The Trustees of Princeton University (US) 2001-06-13 EP claimed
US-6066732-A Process for the preparation of pyrrolo[2,3-d]pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US claimed
WO-2000011004-A1 PROCESS FOR THE PREPARATION OF PYRROLO[2,3-D]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-03-02 WO claimed
EP-0314280-B1 Process for the preparation of fused pyridine compounds UNIV PRINCETON (US) 1996-02-21 EP claimed
US-4895946-A Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1990-01-23 US claimed
EP-0314280-A2 Process for the preparation of fused pyridine compounds THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-05-03 EP claimed