SCHEMBL4661772

SCHEMBL4661772

CC(C)(Br)Cc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.61
TAAR1 Q96RJ0 1/20 0.61
CYP2D6 P10635 2/20 0.56
LMNA P02545 1/20 0.56
TRPA1 O75762 2/20 0.48
CYP1A2 P05177 3/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
ALDH1A1 P00352 3/20 0.46
TSHR P16473 2/20 0.46
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
CALM1 P0DP23 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
FDPS P14324 1/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1B1 Q16678 1/20 0.41
PRMT1 Q99873 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28358439 0.83 SLC6A2 (0.61) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL2313943 0.81 SLC6A2 (0.58) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL7666090 0.81 SLC6A2 (0.58) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL17832229 0.80 SLC6A2 (0.52) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL347187 0.80 SLC6A2 (0.64) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL1572105 0.80 SLC6A2 (0.64) SLC6A2TAAR1CYP2D6LMNATRPA1
Ammonia Solution, Strong SCHEMBL29011215 0.79 SLC6A2 (0.56) SLC6A2TAAR1CYP2D6LMNATRPA1
Ammonia Solution, Strong SCHEMBL10608295 0.78 SLC6A2 (0.61) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL3461269 0.77 SLC6A2 (0.54) SLC6A2TAAR1CYP2D6LMNATRPA1
SCHEMBL4909470 0.77 SLC6A2 (0.67) SLC6A2TAAR1CYP2D6LMNATRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114853686-A Triazole ketone compound and medical application thereof 中国药科大学 2022-08-05 CN disclosed
CN-106588651-B Phenylethylene quaternary carbon compound and preparation method thereof 上海大学 2019-10-11 CN disclosed
CN-106588651-A Styrenic quaternary carbon compound and preparation method thereof 上海大学 2017-04-26 CN disclosed
EP-2004667-A2 NOVEL 11 BETA - HYDROXYANDROSTA-4-ENE-3-ONES Sun Pharma Advanced Research Company Limited (IN) 2008-12-24 EP disclosed
WO-2007099548-A2 NOVEL 11 BETA - HYDROXYANDROSTA-4-ENE-3-ONES SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2007-09-07 WO disclosed
US-4785100-A BROMINATION FOLLOWED BY AMINATION HUELS AKTIENGESELLSHAFT (DE) 1988-11-15 US disclosed
EP-0262348-A2 Process for the preparation of N-substituted morpholine and piperidine derivatives HÜLS AKTIENGESELLSCHAFT (DE) 1988-04-06 EP disclosed