SCHEMBL4662837

SCHEMBL4662837

O=c1[nH]c(=O)n(CCCN2CC3CC3(c3ccc(C(F)(F)F)cc3F)C2)cc1-c1cccnc1F

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 19/20 0.45
KCNH2 Q12809 18/20 0.45
DRD2 P14416 16/20 0.45
DRD4 P21917 1/20 0.45
CYP2C19 P33261 1/20 0.34
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3573467 1.00 DRD3 (0.45) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL15190136 1.00 DRD3 (0.45) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL15190137 1.00 DRD3 (0.45) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL15190064 0.99 DRD3 (0.45) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL3566592 0.90 DRD3 (0.53) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL13314394 0.90 DRD3 (0.53) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL3563042 0.89 DRD3 (0.44) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL3558317 0.89 DRD3 (0.52) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL3559022 0.89 DRD3 (0.52) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL3560097 0.89 DRD3 (0.52) DRD3KCNH2DRD2DRD4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007750-A1 AZABICYCLO [3. 1. 0] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2008-12-31 EP disclosed
WO-2007113232-A1 AZABICYCLO [3. 1. 0] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2007-10-11 WO disclosed