SCHEMBL4662838

SCHEMBL4662838

O=c1[nH]c(=S)ccn1CCCCN1CC2CC2(c2ccc(C(F)(F)F)cc2)C1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 16/20 0.45
KCNH2 Q12809 16/20 0.45
DRD2 P14416 13/20 0.45
CYP1A2 P05177 1/20 0.43
MGLL Q99685 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3554321 1.00 DRD3 (0.45) DRD3KCNH2DRD2CYP1A2MGLL
Hydrochloric Acid SCHEMBL3557043 0.99 DRD3 (0.45) DRD3KCNH2DRD2CYP1A2MGLL
SCHEMBL3570811 0.90 DRD3 (0.49) DRD3KCNH2DRD2CYP1A2
Hydrochloric Acid SCHEMBL3560825 0.89 DRD3 (0.48) DRD3KCNH2DRD2CYP1A2
SCHEMBL3567364 0.88 DRD3 (0.49) DRD3KCNH2DRD2CYP1A2
Hydrochloric Acid SCHEMBL3569370 0.87 DRD3 (0.48) DRD3KCNH2DRD2CYP1A2
SCHEMBL3568192 0.83 DRD3 (0.46) DRD3KCNH2DRD2CYP1A2MGLL
SCHEMBL3566910 0.82 DRD3 (0.49) DRD3KCNH2DRD2CYP1A2
Hydrochloric Acid SCHEMBL3556801 0.82 DRD3 (0.46) DRD3KCNH2DRD2CYP1A2MGLL
SCHEMBL3563967 0.81 DRD3 (0.49) DRD3KCNH2DRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007750-A1 AZABICYCLO [3. 1. 0] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2008-12-31 EP disclosed
WO-2007113232-A1 AZABICYCLO [3. 1. 0] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2007-10-11 WO disclosed