SCHEMBL4665763

SCHEMBL4665763

Cc1ccc(S(=O)(=O)Nc2ccc(Nc3cc(-c4cccc([N+](=O)[O-])c4)ncn3)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 9/20 0.59
CDK9 P50750 9/20 0.59
KMO O15229 1/20 0.54
TNNI3K Q59H18 2/20 0.52
EGFR P00533 1/20 0.52
USP2 O75604 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
TSHR P16473 1/20 0.50
CYP2C19 P33261 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
PLAU P00749 1/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
PLA2G1B P04054 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665854 0.85 BACE1 (0.60) KMOTNNI3KUSP2CYP1A2CYP3A4
SCHEMBL4664257 0.85 CCNT1 (0.64) CCNT1CDK9TNNI3KUSP2CYP1A2
SCHEMBL4109389 0.83 EGFR (0.54) CCNT1CDK9TNNI3KEGFRUSP2
SCHEMBL4667533 0.83 PIM1 (0.59) CCNT1CDK9TNNI3KUSP2CYP1A2
SCHEMBL4665690 0.82 POLB (0.56) TNNI3KUSP2CYP1A2CYP3A4CYP2D6
SCHEMBL4667485 0.82 USP2 (0.54) TNNI3KUSP2CYP1A2CYP3A4CYP2D6
SCHEMBL4664298 0.81 MEN1 (0.51) KMOTNNI3KUSP2CYP1A2CYP3A4
SCHEMBL4664324 0.80 ABL1 (0.55) TNNI3KKDM4EALDH1A1MAPTMEN1
SCHEMBL4098855 0.79 MAPT (0.53) TNNI3KKDM4EALDH1A1MAPTMEN1
SCHEMBL4105292 0.79 HDAC4 (0.49) CCNT1CDK9TNNI3KUSP2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242681-A1 N-4-(6-(Hetero)Aryl-Pyrimidin-4-Ylaminophenyl)-Benzenesulfonamides as Kinase Inhibitors ALTANA PHARMA AG (DE) 2008-10-02 US claimed
EP-1709007-A1 N-4-(6-(HETEO)ARYL-PYRIMIDIN-4-YLAMINOPHENYL)-BENZENESULFONAMIDES AS KINASE INHIBITORS Altana Pharma AG (DE) 2006-10-11 EP claimed
WO-2005070900-A1 N-4-(6- (HETEO) ARYL-PYRIMIDIN-4-YLAMINOPHENYL) -BEZENESULFONAMIDES AS KINASE INHIBITORS ALTANA PHARMA AG (DE) 2005-08-04 WO claimed
US-20080242681-A1 N-4-(6-(Hetero)Aryl-Pyrimidin-4-Ylaminophenyl)-Benzenesulfonamides as Kinase Inhibitors ALTANA PHARMA AG (DE) 2008-10-02 US disclosed
EP-1709007-A1 N-4-(6-(HETEO)ARYL-PYRIMIDIN-4-YLAMINOPHENYL)-BENZENESULFONAMIDES AS KINASE INHIBITORS Altana Pharma AG (DE) 2006-10-11 EP disclosed
WO-2005070900-A1 N-4-(6- (HETEO) ARYL-PYRIMIDIN-4-YLAMINOPHENYL) -BEZENESULFONAMIDES AS KINASE INHIBITORS ALTANA PHARMA AG (DE) 2005-08-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242681-A1 N-4-(6-(Hetero)Aryl-Pyrimidin-4-Ylaminophenyl)-Benzenesulfonamides as Kinase Inhibitors MAP3K19, MAP3K6, MAP3K20 CCNT1 217/4885CDK9 49/4885KMO 915/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.