SCHEMBL4666333

SCHEMBL4666333

Cc1nc(F)ccc1-c1cn(CCCN2CC3CC3(c3ccc(C(F)(F)F)cc3)C2)c(=O)[nH]c1=O

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.48
KCNH2 Q12809 19/20 0.48
DRD2 P14416 16/20 0.48
CYP1A2 P05177 1/20 0.44
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15190297 1.00 DRD3 (0.48) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL15190294 1.00 DRD3 (0.48) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL3561650 1.00 DRD3 (0.48) DRD3KCNH2DRD2CYP1A2DRD4
Hydrochloric Acid SCHEMBL3564771 0.99 DRD3 (0.48) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL3567172 0.92 DRD3 (0.44) DRD3KCNH2DRD2CYP1A2DRD4
Hydrochloric Acid SCHEMBL3566958 0.91 DRD3 (0.44) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL3562135 0.90 KCNH2 (0.48) DRD3KCNH2DRD2CYP1A2
Hydrochloric Acid SCHEMBL3564330 0.89 KCNH2 (0.48) DRD3KCNH2DRD2CYP1A2
SCHEMBL3558310 0.89 DRD3 (0.60) DRD3KCNH2DRD2CYP1A2DRD4
Hydrochloric Acid SCHEMBL3566290 0.88 DRD3 (0.59) DRD3KCNH2DRD2CYP1A2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007750-A1 AZABICYCLO [3. 1. 0] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2008-12-31 EP claimed
WO-2007113232-A1 AZABICYCLO [3. 1. 0] HEXYL DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2007-10-11 WO claimed