SCHEMBL4666903

SCHEMBL4666903

COC[C@H](C)Oc1cc(OC(C)c2ccccc2)cc(C(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GCK P35557 18/20 0.55
RARA P10276 1/20 0.53
RARB P10826 1/20 0.53
RARG P13631 1/20 0.46
LTB4R Q15722 1/20 0.45
LTB4R2 Q9NPC1 1/20 0.45
FFAR1 O14842 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1107734 0.87 GCK (0.57) GCKRARARARBRARG
SCHEMBL12603057 0.87 GCK (0.61) GCKRARARARBRARG
SCHEMBL1107704 0.85 GCK (0.68) GCKRARARARBRARG
SCHEMBL1107456 0.85 GCK (0.68) GCKRARARARBRARG
SCHEMBL2085174 0.85 GCK (0.68) GCKRARARARBRARG
SCHEMBL1107730 0.85 GCK (0.68) GCKRARARARBRARG
SCHEMBL16270273 0.83 GCK (0.57) GCKRARARARBRARG
SCHEMBL1107709 0.83 GCK (0.55) GCKRARARARBRARG
SCHEMBL1107706 0.83 GCK (0.63) GCKRARARARBRARG
SCHEMBL7935638 0.82 GCK (0.83) GCKRARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1992623-A1 Heteroaryl benzamide derivative for use as GLK activator in the treatment of diabetes Astra Zeneca AB (SE) 2008-11-19 EP disclosed