SCHEMBL4667040

SCHEMBL4667040

CCc1cc(-c2cc(Nc3ccc(C)cc3C(=O)OC)n(-c3ccccc3C)n2)ccn1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 9/20 0.42
MAPT P10636 3/20 0.39
TP53 P04637 2/20 0.39
CYP46A1 Q9Y6A2 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
DHODH Q02127 1/20 0.36
NR3C2 P08235 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665900 0.91 ADORA1 (0.51) ADORA1MAPTTP53ADORA3DHODH
SCHEMBL5008775 0.77 ADORA1 (0.55) ADORA1MAPTTP53KDM4EALDH1A1
SCHEMBL5005236 0.76 ADORA1 (0.56) ADORA1MAPTTP53ALDH1A1ADORA3
SCHEMBL5008553 0.76 ADORA1 (0.59) ADORA1MAPTTP53ADORA3DHODH
SCHEMBL3307066 0.75 GFER (0.46) ADORA1MAPTTP53KDM4EALDH1A1
SCHEMBL5005626 0.75 ADORA1 (0.51) ADORA1MAPTALDH1A1ADORA3MAPK13
SCHEMBL5005410 0.75 MAPK14 (0.53) ADORA1KDM4EALDH1A1MAPK13MAPK12
SCHEMBL5005393 0.74 ADORA1 (0.47) ADORA1MAPTTP53KDM4EALDH1A1
SCHEMBL5008431 0.73 ADORA1 (0.62) ADORA1MAPTTP53ADORA3DHODH
SCHEMBL5011998 0.72 MAPT (0.59) ADORA1MAPTTP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed