SCHEMBL4668128

SCHEMBL4668128

CC(=O)NCC(C(=O)Nc1ccccc1)c1ccc(C(=O)Nc2cc(-c3ccsc3)ccc2OC(N)=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 17/20 0.49
HDAC2 Q92769 8/20 0.45
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PLG P00747 1/20 0.39
F7 P08709 1/20 0.39
F3 P13726 1/20 0.39
HDAC3 O15379 5/20 0.38
NCOR2 Q9Y618 2/20 0.38
BCL9 O00512 1/20 0.36
CTNNB1 P35222 1/20 0.36
HDAC4 P56524 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779009 0.88 HDAC1 (0.45) HDAC1HDAC2F2F10PLG
SCHEMBL2685397 0.88 HDAC1 (0.65) HDAC1HDAC2HDAC3NCOR2HDAC4
SCHEMBL4781161 0.87 HDAC1 (0.51) HDAC1HDAC2F2F10PLG
SCHEMBL2686835 0.86 HDAC1 (0.50) HDAC1HDAC2F2F10PLG
SCHEMBL5544366 0.83 HDAC1 (0.45) HDAC1HDAC2F2F10PLG
SCHEMBL2684526 0.81 HDAC1 (0.45) HDAC1HDAC2F2F10PLG
SCHEMBL2685888 0.80 HDAC1 (0.58) HDAC1HDAC2HDAC3NCOR2
SCHEMBL2687859 0.79 HDAC1 (0.66) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL2685976 0.78 HDAC1 (0.44) HDAC1HDAC2F2F10PLG
SCHEMBL2687187 0.77 HDAC1 (0.58) HDAC1HDAC2HDAC3NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-A2 INHIBITORS OF HISTONE DEACETYLASE Merck & Co., Inc. (US) 2008-11-19 EP disclosed
WO-2007100657-A2 INHIBITORS OF HISTONE DEACETYLASE MERCK & CO., INC. (US) 2007-09-07 WO disclosed