SCHEMBL4669199

SCHEMBL4669199

Cc1cnn([C@H]2C[C@H](n3cnc4c(NCC(c5ccccc5)c5ccccc5)nc(NC5CCC(N)CC5)nc43)[C@H](OC(=O)C(F)(F)F)[C@H]2O)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.56
ADORA3 P0DMS8 6/20 0.43
CCNE2 O96020 3/20 0.42
CDK1 P06493 3/20 0.42
CCNE1 P24864 3/20 0.42
CDK2 P24941 3/20 0.42
CCNB2 O95067 2/20 0.42
CDK4 P11802 2/20 0.42
CCNB1 P14635 2/20 0.42
CCND1 P24385 2/20 0.42
CCNB3 Q8WWL7 2/20 0.42
FLT3 P36888 1/20 0.42
CCNA2 P20248 1/20 0.40
CCNA1 P78396 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL590623 1.00 ADORA2A (0.56) ADORA2AADORA3CCNE2CDK1CCNE1
SCHEMBL3153933 1.00 ADORA2A (0.56) ADORA2AADORA3CCNE2CDK1CCNE1
SCHEMBL590622 0.98 ADORA2A (0.56) ADORA2AADORA3CCNE2CDK1CCNE1
SCHEMBL589529 0.93 ADORA2A (0.57) ADORA2AADORA3CCNE2CDK1CCNE1
Trifluoroacetic Acid SCHEMBL590621 0.91 ADORA2A (0.63) ADORA2AADORA3CCNE2CDK1CCNE1
Trifluoroacetic Acid SCHEMBL3153924 0.91 ADORA2A (0.63) ADORA2AADORA3CCNE2CDK1CCNE1
SCHEMBL589528 0.91 ADORA2A (0.57) ADORA2AADORA3CCNE2CDK1CCNE1
SCHEMBL589277 0.89 ADORA2A (0.54) ADORA2AADORA3
SCHEMBL589072 0.87 ADORA2A (0.57) ADORA2AADORA3CCNE2CDK1CCNE1
SCHEMBL589276 0.87 ADORA2A (0.54) ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1841768-B1 PURINE DERIVATIVES ACTING AS A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2008-11-12 EP disclosed