SCHEMBL4669974

SCHEMBL4669974

N#Cc1cc(NCCNc2cnc([N+](=O)[O-])c(-c3ccc(Cl)cc3Cl)n2)ccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.47
GSK3A P49840 4/20 0.41
CDK1 P06493 3/20 0.41
CCNB2 O95067 2/20 0.41
CCNB1 P14635 2/20 0.41
CCNB3 Q8WWL7 2/20 0.41
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
RPS6KB1 P23443 1/20 0.37
CDK2 P24941 1/20 0.37
LIMK1 P53667 1/20 0.37
TAOK1 Q7L7X3 1/20 0.37
SLK Q9H2G2 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
CSNK1G1 Q9HCP0 1/20 0.37
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4670341 0.86 GSK3B (0.63) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL5082188 0.83 GSK3B (0.54) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4675036 0.82 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4672350 0.82 GSK3B (0.51) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4675353 0.80 GSK3B (0.50) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL5076249 0.78 GSK3B (0.62) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4669937 0.78 GSK3B (0.50) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL14175422 0.76 GSK3B (0.64) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL4675401 0.73 IDO1 (0.43) GSK3BGSK3ACDK1CCNB2CCNB1
SCHEMBL5076233 0.72 GSK3B (0.43) GSK3BGSK3ACDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237880-B1 PYRAZINE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2008-01-23 EP disclosed