SCHEMBL4678038

SCHEMBL4678038

C[S+]([O-])c1ccc(C(=O)Nc2cccnc2C(=O)Nc2ncccc2Cl)c(OC2CCC(N)CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 6/20 0.40
PDE4D Q08499 3/20 0.37
SYK P43405 3/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
SCD O00767 5/20 0.36
IRAK1 P51617 1/20 0.36
GAA P10253 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4678044 1.00 IRAK4 (0.40) IRAK4PDE4DSYKPDE4APDE4B
SCHEMBL4268986 0.87 IRAK4 (0.44) IRAK4SYKNPC1RAB9AJAK2
SCHEMBL4268979 0.87 IRAK4 (0.44) IRAK4SYKNPC1RAB9AJAK2
SCHEMBL4278914 0.87 IRAK4 (0.44) IRAK4SYKNPC1RAB9AJAK2
SCHEMBL4279736 0.78 IRAK4 (0.49) IRAK4SYKNPC1RAB9AJAK2
SCHEMBL13608563 0.75 IRAK4 (0.45) IRAK4NPC1RAB9AIRAK1RXFP1
SCHEMBL4276003 0.75 IRAK4 (0.45) IRAK4NPC1RAB9AIRAK1RXFP1
SCHEMBL4269959 0.75 CACNB4 (0.40) IRAK4SYKNPC1RAB9AJAK2
SCHEMBL4272904 0.75 CACNB4 (0.40) IRAK4SYKNPC1RAB9AJAK2
SCHEMBL4269962 0.75 CACNB4 (0.40) IRAK4SYKNPC1RAB9AJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644334-B1 ANTITHROMBOTIC ETHERS LILLY CO ELI (US) 2008-01-02 EP disclosed