SCHEMBL4683036

SCHEMBL4683036

Cc1nc(-c2ccc(C(F)(F)F)cc2)sc1C(N)c1ccsc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
PPARD Q03181 12/20 0.38
PPARA Q07869 7/20 0.38
FFAR1 O14842 3/20 0.38
PPARG P37231 1/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
HSP90AA1 P07900 1/20 0.37
CRHBP P24387 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHR2 Q13324 1/20 0.37
LTA4H P09960 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4678018 0.80 NPC1 (0.46) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL6221868 0.76 NPC1 (0.52) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL5406405 0.76 NPC1 (0.46) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL4854310 0.74 NPC1 (0.50) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL4856478 0.74 NPC1 (0.53) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL4856486 0.74 NPC1 (0.53) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL4854315 0.74 NPC1 (0.50) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL4882934 0.74 NPC1 (0.50) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL3371882 0.74 NPC1 (0.53) NPC1ALDH1A1GAAPPARDPPARA
SCHEMBL27650489 0.74 NPC1 (0.56) NPC1ALDH1A1GAAPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1513796-B1 PHENYLOXYALKANOIC ACID DERIVATIVES AS HPPAR ACTIVATORS SMITHKLINE BEECHAM CORP (US) 2008-02-13 EP disclosed