SCHEMBL4684152

SCHEMBL4684152

CC1CC1CN(Cc1ccccc1)c1cc(-c2nnc(C(C)(CNC(=O)O)c3ccccc3)o2)cc(N(C)S(C)(=O)=O)n1

nearest known ligand 0.42

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.42
BACE2 Q9Y5Z0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4946005 0.86 BACE1 (0.43) BACE1BACE2
SCHEMBL2023415 0.86 BACE1 (0.43) BACE1BACE2
SCHEMBL2018791 0.83 BACE1 (0.43) BACE1BACE2
SCHEMBL2018789 0.83 BACE1 (0.43) BACE1BACE2
SCHEMBL2024027 0.83 BACE1 (0.53) BACE1BACE2
SCHEMBL2023745 0.83 BACE1 (0.53) BACE1BACE2
SCHEMBL12578958 0.80 BACE1 (0.49) BACE1BACE2
SCHEMBL5650748 0.78 BACE1 (0.40) BACE1BACE2
SCHEMBL4946010 0.78 BACE1 (0.42) BACE1BACE2
SCHEMBL5651224 0.77 BACE1 (0.49) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740581-A4 2, 4, 6-SUBSTITUTED PYRIDYL DERIVATIVE COMPOUNDS USEFUL AS BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO INC (US) 2008-01-23 EP disclosed
EP-1740581-A1 2, 4, 6-SUBSTITUTED PYRIDYL DERIVATIVE COMPOUNDS USEFUL AS BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER\"S DISEASE Merck and Co., Inc. (US) 2007-01-10 EP disclosed
WO-2005103043-A1 2, 4, 6-SUBSTITUTED PYRIDYL DERIVATIVE COMPOUNDS USEFUL AS BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER’S DISEASE MERCK & CO., INC. (US) 2005-11-03 WO disclosed