SCHEMBL4686783

SCHEMBL4686783

COc1cc(CCC(=O)c2sc(C)c3c2C[C@@H]2C3C2(C)C)cc(Cl)c1OC[C@@H](O)CO

nearest known ligand 0.77

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.77
S1PR3 Q99500 15/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2943713 1.00 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL2948296 1.00 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL4687053 0.94 S1PR1 (0.82) S1PR1S1PR3
SCHEMBL2943701 0.94 S1PR1 (0.84) S1PR1S1PR3
SCHEMBL2942033 0.94 S1PR1 (0.84) S1PR1S1PR3
SCHEMBL2947649 0.91 S1PR1 (0.89) S1PR1S1PR3
SCHEMBL2943026 0.91 S1PR1 (0.89) S1PR1S1PR3
SCHEMBL2949102 0.91 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL2944348 0.91 S1PR1 (0.77) S1PR1S1PR3
SCHEMBL2455849 0.91 S1PR1 (0.79) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805163-B1 1,1A,5,5A-TETRAHYDRO-3-THIA-CYCLOPROPA[A]PENTALENES: TRICYCLIC THIOPHENE DERIVATIVES AS S1P1/EDG1 RECEPTOR AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2008-10-01 EP disclosed