SCHEMBL4687680

SCHEMBL4687680

Cc1cc(CNC(=O)Oc2sc(C)c3c2C[C@@H]2[C@H]3C2(C)C)cc(C)c1OCC(CO)CO

nearest known ligand 0.67

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.67
S1PR3 Q99500 18/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688456 0.93 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL4689663 0.93 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL4687690 0.89 S1PR1 (0.65) S1PR1S1PR3
SCHEMBL4690803 0.89 S1PR1 (0.65) S1PR1S1PR3
SCHEMBL2942937 0.87 S1PR1 (0.76) S1PR1S1PR3
SCHEMBL4689440 0.87 S1PR1 (0.59) S1PR1S1PR3
SCHEMBL4688452 0.82 S1PR1 (0.55) S1PR1S1PR3
SCHEMBL4686610 0.82 S1PR1 (0.55) S1PR1S1PR3
SCHEMBL4690884 0.81 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL2950882 0.80 S1PR1 (1.00) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805163-B1 1,1A,5,5A-TETRAHYDRO-3-THIA-CYCLOPROPA[A]PENTALENES: TRICYCLIC THIOPHENE DERIVATIVES AS S1P1/EDG1 RECEPTOR AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2008-10-01 EP claimed