SCHEMBL4688407

SCHEMBL4688407

COc1ccc2c(=O)n(C)c(CN(C(C)C)C(C)C)c(-c3ccccc3)c2c1

nearest known ligand 0.77

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.77
KCNH2 Q12809 2/20 0.77
DPP4 P27487 5/20 0.59
TACR1 P25103 6/20 0.52
MAPK8 P45983 1/20 0.47
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689161 0.90 KCNA5 (0.79) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL4686913 0.87 KCNA5 (1.00) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL4686242 0.86 KCNA5 (0.81) KCNA5KCNH2DPP4TACR1MAPK8
Hydrochloric Acid SCHEMBL295443 0.86 KCNA5 (0.98) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL4685992 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL1381998 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL2904903 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL3115349 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL1382996 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4TACR1MAPK8
SCHEMBL14303480 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4TACR1MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322619-B1 ISOQUINOLINONE POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2008-01-23 EP disclosed
US-6870055-B2 Isoquinolinone potassium channels inhibitors MERCK & CO., INC. (US) 2005-03-22 US disclosed