SCHEMBL4688684

SCHEMBL4688684

CC(c1ccc(Cl)cc1)C(CNC(=O)C(C)(C)Oc1cccnc1)c1ccc(Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.62
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
CNR2 P34972 9/20 0.48
ALOX15 P16050 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691697 0.97 CNR1 (0.67) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL2653184 0.93 CNR1 (0.56) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4688895 0.90 CNR1 (0.54) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4690815 0.89 CNR1 (0.53) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4688372 0.89 CNR1 (0.54) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4691778 0.87 CNR1 (0.58) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4688836 0.87 CNR1 (0.60) CNR1CNR2
SCHEMBL4689273 0.87 CNR1 (0.55) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4690920 0.87 CNR1 (0.51) CNR1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4693315 0.86 CYP1A2 (0.56) CNR1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed