SCHEMBL4690913

SCHEMBL4690913

COc1ccc2c(=O)n(C)c(N)c(-c3ccccc3)c2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.66
KCNH2 Q12809 2/20 0.66
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
CRHBP P24387 1/20 0.55
CRHR2 Q13324 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
DPP4 P27487 4/20 0.55
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
MAPK8 P45983 1/20 0.51
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
HPGD P15428 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
BRD4 O60885 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3118253 0.86 KCNA5 (0.69) KCNA5KCNH2MEN1KMT2ADPP4
SCHEMBL4685992 0.83 KCNA5 (0.76) KCNA5KCNH2DPP4CA1CA2
SCHEMBL4685991 0.82 KCNA5 (0.61) KCNA5KCNH2DPP4CA1CA2
SCHEMBL3094005 0.82 KCNA5 (0.63) KCNA5KCNH2DPP4CA1CA2
SCHEMBL2900202 0.81 KCNA5 (0.73) KCNA5KCNH2DPP4CA1CA2
SCHEMBL3616349 0.81 KCNA5 (0.64) KCNA5KCNH2MEN1KMT2ADPP4
SCHEMBL1382996 0.81 KCNA5 (0.76) KCNA5KCNH2DPP4CA1CA2
SCHEMBL3115349 0.81 KCNA5 (0.76) KCNA5KCNH2DPP4CA1CA2
SCHEMBL1381998 0.81 KCNA5 (0.76) KCNA5KCNH2MEN1KMT2ADPP4
SCHEMBL2904903 0.81 KCNA5 (0.76) KCNA5KCNH2DPP4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322619-B1 ISOQUINOLINONE POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2008-01-23 EP disclosed
US-6870055-B2 Isoquinolinone potassium channels inhibitors MERCK & CO., INC. (US) 2005-03-22 US disclosed