SCHEMBL4692413

SCHEMBL4692413

Cc1cccc(C)c1C(=O)N1CC2CN(c3cccc(CCC(N)=O)c3)CC2C1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.53
HCRTR2 O43614 12/20 0.53
KCNH2 Q12809 1/20 0.43
CCR5 P51681 6/20 0.41
PLA2G10 O15496 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231170 0.95 HCRTR1 (0.52) HCRTR1HCRTR2KCNH2CCR5PLA2G10
SCHEMBL5236364 0.94 HCRTR1 (0.47) HCRTR1HCRTR2KCNH2CCR5PLA2G10
SCHEMBL5237741 0.92 HCRTR1 (0.44) HCRTR1HCRTR2KCNH2CCR5PLA2G10
SCHEMBL5238954 0.90 HCRTR1 (0.43) HCRTR1HCRTR2CCR5PLA2G10
SCHEMBL5231850 0.90 HCRTR1 (0.43) HCRTR1HCRTR2KCNH2CCR5PLA2G10
SCHEMBL5235800 0.89 HCRTR1 (0.44) HCRTR1HCRTR2KCNH2CCR5
SCHEMBL5234579 0.89 HCRTR1 (0.42) HCRTR1HCRTR2KCNH2PLA2G10
SCHEMBL5239352 0.89 HCRTR1 (0.55) HCRTR1HCRTR2PLA2G10
SCHEMBL5237249 0.88 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL4968486 0.88 HCRTR1 (0.42) HCRTR1HCRTR2KCNH2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed