SCHEMBL4692776

SCHEMBL4692776

COc1ccccc1/C(Br)=C(\NC(=O)c1ccccc1)C(=O)N1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
NPC1 O15118 4/20 0.48
RAB9A P51151 3/20 0.48
HPGD P15428 2/20 0.47
HTT P42858 2/20 0.47
KMT2A Q03164 4/20 0.46
ALDH1A1 P00352 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CYP2C9 P11712 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
MAPT P10636 2/20 0.45
AHR P35869 1/20 0.45
GFER P55789 1/20 0.45
ALOX15 P16050 1/20 0.44
MAPK1 P28482 2/20 0.43
ALOX5 P09917 1/20 0.43
KCNK3 O14649 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43
PKM P14618 1/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692778 1.00 GAA (0.49) GAANPC1RAB9AHPGDHTT
SCHEMBL4744757 0.92 TSHR (0.53) GAANPC1RAB9AHPGDHTT
SCHEMBL4744761 0.92 TSHR (0.53) GAANPC1RAB9AHPGDHTT
SCHEMBL4688665 0.88 MAPT (0.50) GAARAB9AHPGDHTTKMT2A
SCHEMBL5896804 0.88 MAPT (0.50) GAARAB9AHPGDHTTKMT2A
SCHEMBL5896791 0.88 MAPT (0.50) GAARAB9AHPGDHTTKMT2A
SCHEMBL29385179 0.88 MAPT (0.50) GAARAB9AHPGDHTTKMT2A
SCHEMBL4745685 0.87 MAPT (0.48) GAARAB9AHPGDHTTKMT2A
SCHEMBL4745679 0.87 MAPT (0.48) GAARAB9AHPGDHTTKMT2A
SCHEMBL4747319 0.84 GAA (0.52) GAANPC1RAB9AHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581496-A4 2-SUBSTITUTED-3-PROPENAMIDE DERIVATIVES AND METHODS OF USING THE SAME GILEAD SCIENCES INC (US) 2008-04-23 EP disclosed
EP-1581496-A2 2-SUBSTITUTED-3-PROPENAMIDE DERIVATIVES AND METHODS OF USING THE SAME GILEAD SCIENCES, INC. (US) 2005-10-05 EP disclosed
WO-2004050613-A2 2-SUBSTITUTED-3-PROPENAMIDE DERIVATIVES AND METHODS OF USING THE SAME GILEAD SCIENCES, INC. (US) 2004-06-17 WO disclosed