SCHEMBL4692850

SCHEMBL4692850

CC(c1ccc(Cl)cc1)C(CNC(=O)C(C)(C)Oc1ccc(C(F)(F)F)cn1)c1cc(F)cc(C#N)c1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 0.62
CNR2 P34972 7/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
KCNH2 Q12809 1/20 0.60
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689154 0.94 CNR1 (0.65) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL5153055 0.93 CNR1 (0.63) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2170495 0.91 CNR1 (0.72) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3668309 0.91 CNR1 (0.72) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2652272 0.91 CNR1 (0.60) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL1567733 0.91 CNR1 (0.72) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL5148428 0.90 CNR1 (0.75) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4691565 0.88 CNR1 (0.58) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4692291 0.87 CNR1 (0.53) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4688432 0.87 CNR1 (0.59) CNR1CNR2CYP2D6CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed