SCHEMBL4693569

SCHEMBL4693569

COc1ccc(NC2=C(c3ccccc3)C(=O)N(Cc3ccc(C(=O)O)cc3)C2=O)cc1

nearest known ligand 0.81

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 8/20 0.81
NR1H3 Q13133 8/20 0.81
GSK3B P49841 2/20 0.49
MAPT P10636 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CASP3 P42574 1/20 0.46
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44
ACP1 P24666 1/20 0.44
MAOA P21397 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
AKR1C3 P42330 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688675 0.93 NR1H2 (0.80) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4450601 0.90 NR1H2 (1.00) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4692898 0.85 NR1H2 (0.81) NR1H2NR1H3MAPTSMN1; SMN2CASP3
SCHEMBL4686588 0.85 NR1H2 (0.85) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4691707 0.82 NR1H2 (0.76) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4688601 0.81 NR1H2 (0.78) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4685907 0.81 NR1H2 (1.00) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4690915 0.81 NR1H2 (0.73) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4684030 0.80 NR1H2 (0.80) NR1H2NR1H3GSK3BMAPTSMN1; SMN2
SCHEMBL4688066 0.80 NR1H2 (0.80) NR1H2NR1H3MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646626-B1 PYRROLE-2, 5-DIONE DERIVATIVES AS LIVER X RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2008-07-02 EP claimed