SCHEMBL4694081

SCHEMBL4694081

CC(c1ccc(F)cc1)C(CNC(=O)C(C)(C)Oc1ccc(C(F)(F)F)cn1)c1cc(F)cc(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 13/20 0.51
CNR2 P34972 3/20 0.45
CYP2C9 P11712 2/20 0.42
CYP2D6 P10635 1/20 0.42
KCNH2 Q12809 1/20 0.42
DGAT2 Q96PD7 1/20 0.40
SCN9A Q15858 4/20 0.36
LMNA P02545 1/20 0.35
CYP2C19 P33261 1/20 0.35
EPHX2 P34913 1/20 0.35
CYP2J2 P51589 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691565 0.94 CNR1 (0.58) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL4788252 0.92 CNR1 (0.49) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL4689154 0.88 CNR1 (0.65) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL4692012 0.85 CNR1 (0.41) CNR1CNR2EPHX2
SCHEMBL4690869 0.84 CNR1 (0.71) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL4688614 0.84 CNR1 (0.58) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL4688432 0.83 CNR1 (0.59) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL4692291 0.83 CNR1 (0.53) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL3371233 0.83 CNR1 (0.72) CNR1CNR2CYP2C9CYP2D6KCNH2
SCHEMBL2653109 0.83 CNR1 (0.62) CNR1CNR2CYP2C9CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed