SCHEMBL4694454

SCHEMBL4694454

CC(c1ccc(Cl)cc1)C(CNC(=O)C(C)(C)Oc1cc(C(F)(F)F)ccn1)c1cncc(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.47
DGAT2 Q96PD7 1/20 0.42
CNR2 P34972 6/20 0.41
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
KCNH2 Q12809 1/20 0.39
CCR5 P51681 2/20 0.36
P2RX3 P56373 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688614 0.90 CNR1 (0.58) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL4691581 0.88 CNR1 (0.48) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL4691568 0.87 CNR1 (0.43) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2653600 0.87 CNR1 (0.52) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL4692090 0.84 CNR1 (0.47) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL3374861 0.83 CNR1 (0.67) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4788252 0.82 CNR1 (0.49) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL1571723 0.82 CNR1 (0.55) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL2653127 0.81 CNR1 (0.53) CNR1DGAT2CNR2CYP2D6CYP2C9
SCHEMBL4692291 0.81 CNR1 (0.53) CNR1DGAT2CNR2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed