SCHEMBL4694633

SCHEMBL4694633

CC(C1CCC1)C(CNC(=O)C(C)(C)Oc1ccncc1C(F)(F)F)c1cncc(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 4/20 0.41
P2RX7 Q99572 1/20 0.34
GAA P10253 1/20 0.33
PTGES O14684 3/20 0.33
PTGS2 P35354 3/20 0.33
CCR5 P51681 2/20 0.33
CNR1 P21554 3/20 0.33
CNR2 P34972 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689785 0.84 CNR1 (0.37) SSTR4CNR1CNR2
SCHEMBL4692580 0.84 ACACB (0.35) PTGESPTGS2CCR5CNR1CNR2
SCHEMBL3371182 0.83 CNR1 (0.40) SSTR4CNR1CNR2
SCHEMBL3370475 0.79 CNR1 (0.44) CNR1CNR2
SCHEMBL3369677 0.77 ACACB (0.34) CCR5CNR1CNR2
SCHEMBL3371801 0.75 CNR1 (0.56) CNR1CNR2
SCHEMBL4689257 0.69 CNR1 (0.39) CNR1CNR2
SCHEMBL4688390 0.69 CNR1 (0.36) CNR1CNR2
SCHEMBL1571723 0.68 CNR1 (0.55) CNR1CNR2
SCHEMBL4688592 0.68 CNR1 (0.40) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed