SCHEMBL469610

SCHEMBL469610

CC(C)(Br)CC(C)(C)CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.55
ALDH1A1 P00352 1/20 0.47
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9625482 0.87 CHRM2 (0.63) CHRM2ALDH1A1MEN1CYP1A2CYP2C19
SCHEMBL2599276 0.84 CHRM2 (0.56) CHRM2ALDH1A1MEN1CYP1A2CYP2C19
SCHEMBL799700 0.81 CHRM2 (0.58) CHRM2ALDH1A1MEN1CYP1A2CYP2C19
SCHEMBL3727196 0.80 CHRM2 (0.56) CHRM2ALDH1A1
SCHEMBL5962347 0.79 CHRM2 (0.54) CHRM2ALDH1A1MEN1CYP1A2CYP2C19
SCHEMBL19228128 0.79 CHRM2 (0.55) CHRM2ALDH1A1
SCHEMBL14481161 0.77 CHRM2 (0.54) CHRM2ALDH1A1
SCHEMBL7260725 0.77 CHRM2 (0.54) CHRM2ALDH1A1
SCHEMBL14480981 0.77 CHRM2 (0.54) CHRM2ALDH1A1
SCHEMBL7286379 0.77 CHRM2 (0.53) CHRM2ALDH1A1MEN1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012034116-A2 SMALL MOLECULES AS EPIGENETIC MODULATORS OF LYSINE-SPECIFIC DEMETHYLASE 1 AND METHODS OF TREATING DISORDERS THE JOHNS HOPKINS UNIVERSITY (US) 2012-03-15 WO disclosed