SCHEMBL469670

SCHEMBL469670

C[Si](C)(C)OC[C@@H]1C[C@H](O[Si](C)(C)C)CC(=O)O1

nearest known ligand 0.38

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22077666 1.00 SMN1; SMN2 (0.31) SMN1; SMN2
SCHEMBL13074797 0.84 CYP1A2 (0.30)
SCHEMBL10212414 0.82
SCHEMBL13260909 0.80 HMGCR (0.41)
SCHEMBL9287478 0.79 TOP2A (0.39)
SCHEMBL19676622 0.74 SMN1; SMN2 (0.52) SMN1; SMN2
SCHEMBL10328064 0.73
SCHEMBL7952252 0.73
SCHEMBL19493420 0.73
SCHEMBL18536367 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200606-B1 PROCESS FOR THE PREPARATION OF COMPOUNDS USEFUL AS INHIBITORS OF SGLT JANSSEN PHARMACEUTICA NV (BE) 2017-10-25 EP disclosed
EP-3133071-A1 C-ARYL INDICAN DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR AND USES THEREOF Shanghai De Novo Pharmatech Co Ltd. (CN) 2017-02-22 EP disclosed
EP-2324002-B1 PROCESSES FOR THE PREPARATION OF SGLT2 INHIBITORS THERACOS SUB LLC (US) 2016-10-05 EP disclosed
WO-2016070740-A1 A CLASS OF NEW TYPE SGLT2 INHIBITOR COMPOUND AND A PHARMACEUTICAL COMPOSITION THEREOF 镇江新元素医药科技有限公司 2016-05-12 WO disclosed
WO-2015132803-A2 PROCESS FOR THE PREPARATION OF (1S)-1,5-ANHYDRO-1-C-[4-CHLORO-3-[(4-ETHOXYPHENYL)METHYL]PHENYL]-D-GLUCITOL AND ITS SOLVATE THEREOF MSN LABORATORIES PRIVATE LIMITED (IN) 2015-09-11 WO disclosed
US-8575321-B2 Benzylbenzene derivatives and methods of use THERACOS, INC. (US) 2013-11-05 US disclosed
US-20120329732-A1 BENZYLBENZENE DERIVATIVES AND METHODS OF USE THERACOS, INC. (US) 2012-12-27 US disclosed
WO-2012165914-A2 NOVEL DIPHENYLMETHANE DERIVATIVES AS SGLT2 INHIBITORS GREEN CROSS CORPORATION (KR) 2012-12-06 WO disclosed
WO-2012033390-A2 NOVEL THIOPHENE DERIVATIVE AS SGLT2 INHIBITOR AND PHARMACEUTICAL COMPOSITION COMPRISING SAME GREEN CROSS CORPORATION (KR) 2012-03-15 WO disclosed
US-8106021-B2 Benzylbenzene derivatives and methods of use THERACOS, INC. (US) 2012-01-31 US disclosed
US-20110207661-A1 BENZYLBENZENE DERIVATIVES AND METHODS OF USE THERACOS, INC. (US) 2011-08-25 US disclosed
WO-2011048112-A1 GLYCOSIDE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2011-04-28 WO disclosed
US-7838499-B2 Benzylbenzene derivatives and methods of use THERACOS, INC. (US) 2010-11-23 US disclosed
US-7803778-B2 Glucose transport inhibitors and methods of use THERACOS, INC. (US) 2010-09-28 US disclosed
WO-2010022313-A2 PROCESSES FOR THE PREPARATION OF SGLT2 INHIBITORS THERACOS, INC. (US) 2010-02-25 WO disclosed
WO-2010009243-A1 DEUTERATED BENZYLBENZENE DERIVATIVES AND METHODS OF USE THERACOS, INC. (US) 2010-01-21 WO disclosed
US-20090118201-A1 BENZYLBENZENE DERIVATIVES AND METHODS OF USE THERACOSBIO, LLC 2009-05-07 US disclosed
US-20070275907-A1 GLUCOSE TRANSPORT INHIBITORS AND METHODS OF USE SEED, BRIAN 2007-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110207661-A1 BENZYLBENZENE DERIVATIVES AND METHODS OF USE SLC5A2, SLC5A1, SLC2A4 SMN1; SMN2 3758/4885
US-20090118201-A1 BENZYLBENZENE DERIVATIVES AND METHODS OF USE SLC5A2, SLC5A1, SLC2A4 SMN1; SMN2 3758/4885
US-20120329732-A1 BENZYLBENZENE DERIVATIVES AND METHODS OF USE SLC5A2, SLC5A1, SLC2A4 SMN1; SMN2 3758/4885
US-20070275907-A1 GLUCOSE TRANSPORT INHIBITORS AND METHODS OF USE SLC5A1, SLC5A2, SLC2A1 SMN1; SMN2 3754/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.