SCHEMBL4696887

SCHEMBL4696887

NC(=O)n1ncc2c1C(C(=O)O)N1C[C@H]2N(OCc2ccccc2)C1=O

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 3/20 0.33
CYP2C19 P33261 2/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
DHFR P00374 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30
PREP P48147 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696891 1.00 KCNA5 (0.33) KCNA5CYP2C19POLBCYP3A4CYP2C9
SCHEMBL4131490 0.91 KCNA5 (0.33) KCNA5CYP2C19POLBCYP3A4CYP2C9
SCHEMBL4131485 0.91 KCNA5 (0.33) KCNA5CYP2C19POLBCYP3A4CYP2C9
SCHEMBL4131495 0.91 KCNA5 (0.33) KCNA5CYP2C19POLBCYP3A4CYP2C9
SCHEMBL4695568 0.87 GRIN2B (0.35) KCNA5
SCHEMBL4695565 0.87 GRIN2B (0.35) KCNA5
SCHEMBL4695570 0.87 GRIN2B (0.35) KCNA5
SCHEMBL2066952 0.86 KCNA5 (0.36) KCNA5CYP2C19POLBCYP3A4CYP2C9
SCHEMBL20557817 0.86 KCNA5 (0.36) KCNA5CYP2C19POLBCYP3A4CYP2C9
SCHEMBL4142823 0.85 TSHR (0.37) KCNA5CYP2C19POLBCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed