SCHEMBL4697400

SCHEMBL4697400

CN1CC2CCN(c3ccc(N4CCN(c5cnccn5)CC4)cc3)C2C1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 15/20 0.54
GPR119 Q8TDV5 1/20 0.54
KCNH2 Q12809 4/20 0.48
DRD2 P14416 2/20 0.44
DRD3 P35462 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063131 1.00 HRH3 (0.54) HRH3GPR119KCNH2DRD2DRD3
SCHEMBL3061109 0.86 HRH3 (0.61) HRH3GPR119KCNH2
SCHEMBL3058263 0.84 HRH3 (0.63) HRH3KCNH2DRD2DRD3
SCHEMBL3062935 0.82 HRH3 (0.60) HRH3KCNH2DRD2DRD3
SCHEMBL3048621 0.81 HRH3 (0.60) HRH3GPR119KCNH2
SCHEMBL3060025 0.79 HRH3 (0.66) HRH3GPR119KCNH2
SCHEMBL3060029 0.79 HRH3 (0.66) HRH3GPR119KCNH2
SCHEMBL3067701 0.78 HRH3 (0.55) HRH3GPR119KCNH2
SCHEMBL3057757 0.77 HRH3 (0.54) HRH3KCNH2DRD2DRD3
SCHEMBL3065520 0.77 HRH3 (0.54) HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001885-A2 OCTAHYDRO-PYRROLO[3,4-B]PYRROLE DERIVATIVES Abbott Laboratories (US) 2008-12-17 EP claimed
WO-2007100990-A2 OCTAHYDRO-PYRROLO[3,4-B] PYRROLE DERIVATIVES AND THEIR USE AS HISTAMINE-3 RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2007-09-07 WO claimed