SCHEMBL4697982

SCHEMBL4697982

CC1(c2cccc(C3(NCC(O)C(Cc4cc(F)cc(F)c4)NC(=O)O)CC3)c2)CCCO1

nearest known ligand 0.89

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.89
CTSD P07339 11/20 0.62
CYP3A4 P08684 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4698235 0.94 BACE1 (1.00) BACE1CTSDCYP3A4
SCHEMBL5578973 0.89 BACE1 (0.84) BACE1CTSDCYP3A4
SCHEMBL4702961 0.85 BACE1 (0.75) BACE1CTSDCYP3A4
SCHEMBL6701304 0.85 BACE1 (0.68) BACE1CTSDCYP3A4
SCHEMBL6701309 0.85 BACE1 (0.68) BACE1CTSDCYP3A4
SCHEMBL4819310 0.84 BACE1 (0.64) BACE1CTSDCYP3A4
SCHEMBL3355039 0.83 BACE1 (0.78) BACE1CTSDCYP3A4
SCHEMBL3355037 0.83 BACE1 (0.78) BACE1CTSDCYP3A4
SCHEMBL4819302 0.83 BACE1 (0.69) BACE1CTSDCYP3A4
SCHEMBL5579109 0.82 BACE1 (0.86) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937638-A1 METHODS OF TREATING AMYLOIDOSIS USING ARYL-CYCLOPROPYL DERIVATIVE ASPARTYL PROTEASE INHIBITORS Elan Pharmaceuticals Inc. (US) 2008-07-02 EP disclosed
WO-2007047306-A1 METHODS OF TREATING AMYLOIDOSIS USING ARYL-CYCLOPROPYL DERIVATIVE ASPARTYL PROTEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 2007-04-26 WO disclosed