SCHEMBL469805

SCHEMBL469805

CC(C)c1ccc(NC(=S)N/N=C2\C(=O)Nc3ccccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.47
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
IGF1R P08069 1/20 0.44
PDGFRB P09619 1/20 0.44
GLB1 P16278 1/20 0.44
CTRC Q99895 1/20 0.44
MAPT P10636 4/20 0.44
TDP1 Q9NUW8 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 2/20 0.44
SLC2A1 P11166 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 2/20 0.43
ALOX12 P18054 2/20 0.43
HPGD P15428 1/20 0.43
GPR55 Q9Y2T6 1/20 0.43
CA12 O43570 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10085722 0.87 KDR (0.61) KDRMAPTALDH1A1CA12CA1
SCHEMBL469802 0.87 MAPT (0.51) KDRMAPTTDP1MEN1KMT2A
SCHEMBL469854 0.87 KDR (0.56) KDRMAPTMEN1KMT2APOLB
SCHEMBL18974340 0.85 KDR (0.49) KDRMAPTMEN1KMT2APOLB
SCHEMBL10084866 0.85 LRRK2 (0.53) KDRMAPTKMT2AALDH1A1GAA
SCHEMBL31491999 0.85 LRRK2 (0.53) KDRMAPTKMT2AALDH1A1GAA
SCHEMBL470031 0.84 MAPT (0.56) KDRMAPTTDP1MEN1KMT2A
SCHEMBL14075826 0.84 MAPT (0.56) KDRMAPTTDP1MEN1KMT2A
SCHEMBL469876 0.84 KDR (0.46) KDRMAPTTDP1MEN1KMT2A
SCHEMBL455695 0.84 SLC2A1 (0.44) EGFRERBB2IGF1RPDGFRBGLB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033601-A1 THIOSEMICARBAZONES WITH MDR1 - INVERSE ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2012-03-15 WO disclosed