SCHEMBL4698377

SCHEMBL4698377

NN(C(=O)c1ccc(NC(=O)OC2CCN(CI)C2)cc1)c1cccc(-c2cccs2)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
CHRM4 P08173 1/20 0.39
DRD4 P21917 11/20 0.39
DRD2 P14416 10/20 0.39
HTR2A P28223 9/20 0.39
MCHR1 Q99705 1/20 0.39
RHOA P61586 1/20 0.39
HDAC3 O15379 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
BCHE P06276 2/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4578951 0.88 HDAC1 (0.44) HDAC1HDAC2CHRM4MCHR1RHOA
SCHEMBL4579158 0.86 HDAC1 (0.45) HDAC1HDAC2MCHR1RHOAHDAC3
SCHEMBL4579949 0.79 HDAC1 (0.41) HDAC1HDAC2MCHR1HDAC3
SCHEMBL4578187 0.79 HDAC1 (0.44) HDAC1HDAC2HDAC3
SCHEMBL4579714 0.77 HDAC1 (0.44) HDAC1HDAC2HDAC3
SCHEMBL4578792 0.77 HDAC1 (0.48) HDAC1HDAC2HDAC3
SCHEMBL4579958 0.75 HDAC1 (0.61) HDAC1HDAC2HDAC3
SCHEMBL4578547 0.73 HDAC1 (0.43) HDAC1HDAC2HDAC3BCHE
SCHEMBL4579959 0.72 HDAC1 (0.41) HDAC1HDAC2HDAC3
SCHEMBL4580090 0.72 HDAC1 (0.59) HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007720-A1 BENZAMIDE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2008-12-31 EP disclosed
WO-2007118137-A1 BENZAMIDE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2007-10-18 WO disclosed