SCHEMBL469850

SCHEMBL469850

C=CN(C)/C=C\N

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517100 0.71
SCHEMBL13384114 0.71
SCHEMBL16790337 0.69
Ammonia Solution, Strong SCHEMBL7051004 0.68
Hydrochloric Acid SCHEMBL10572428 0.68
SCHEMBL4933531 0.67
Formamide SCHEMBL27593949 0.67
SCHEMBL4441677 0.67
SCHEMBL1021476 0.65
SCHEMBL757803 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024008967-A1 LIPID NANOPARTICLES COMPRISING AN IMIDAZOLIUM-BASED CATIONIC LIPID POLYPLUS TRANSFECTION (FR) 2024-01-11 WO disclosed
US-20230304002-A1 TRANSTHYRETIN (TTR) iRNA COMPOSITIONS AND METHODS OF USE THEREOF FOR TREATING OR PREVENTING TTR-ASSOCIATED OCULAR DISEASES BANK OF AMERICA, N.A. 2023-09-28 US disclosed
US-11589583-B2 Pyrrolidinones herbicides FMC CORPORATION (US) 2023-02-28 US disclosed
WO-2023009785-A1 TEAD INHIBITORS AND USES THEREOF CEDILLA THERAPEUTICS, INC. (US) 2023-02-02 WO disclosed
WO-2022188819-A1 SOS1 PROTEOLYSIS MODULATOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 苏州泽璟生物制药股份有限公司 2022-09-15 WO disclosed
US-20220030863-A9 PYRROLIDINONES HERBICIDES FMC CORPORATION 2022-02-03 US disclosed
EP-3359154-B1 WNT SIGNALING PATHWAY INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF Suzhou Yunxuan Yiyao Keji Youxian Gongsi (CN) 2021-05-26 EP disclosed
US-20200367494-A1 PYRROLIDINONES HERBICIDES FMC CORP (US) 2020-11-26 US disclosed
WO-2020192280-A1 DOUBLE BASIC-FUNCTIONALIZED IONIC LIQUID WITH SURFACE ACTIVITY AND PREPARATION METHOD THEREFOR 枣庄学院 2020-10-01 WO disclosed
EP-3549933-A1 HETEROCYCLIC COMPOUND, AND ARTHROPOD PEST CONTROL COMPOSITION CONTAINING SAME Sumitomo Chemical Company, Limited (JP) 2019-10-09 EP disclosed
US-20160028016-A1 BORON-NITROGEN POLYAROMATIC COMPOUNDS AND THEIR USE IN OLEDS UNIVERSAL DISPLAY CORPORATION (US) 2016-01-28 US disclosed
US-20140340820-A1 CONDUCTIVE MATERIAL FORMULATION AND USE THEREOF ETERNAL CHEMICAL CO., LTD. (TW) 2014-11-20 US disclosed
EP-2529733-A1 Antibacterial combination therapy E-Therapeutics Plc (GB) 2012-12-05 EP disclosed
US-20120122679-A1 MESOIONIC PESTICIDES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-05-17 US disclosed
WO-2012033800-A1 COMPOSITION AND METHOD FOR INHIBITING PREMATURE POLYMERIZATION GENERAL ELECTRIC COMPANY (US) 2012-03-15 WO disclosed
US-20110009638-A1 METHOD FOR PREPARING 3-TRIFLUOROMETHYL CHALCONES E.I. DU PONT DE NEMOURS AND COMPANY (DE) 2011-01-13 US disclosed
WO-2010109185-A2 PROCESS FOR THE PREPARATION OF DOXAZOSIN AND SALTS THEREOF CIPLA LIMITED (IN) 2010-09-30 WO disclosed
EP-0906257-B2 MIXTURES CONTAINING MONOMERS AND STABILIZERS BASF SE (DE) 2010-04-07 EP disclosed
EP-2044169-B1 USE OF PT- AND PD-BIS- AND TETRA-CARBON COMPLEXES WITH BRIDGED CARBON LIGANDS IN OLEDS BASF SE (DE) 2009-11-25 EP disclosed
EP-0885180-B1 STABILIZED MONOMER COMPOSITION BASF AG (DE) 2007-04-11 EP disclosed