SCHEMBL4698581

SCHEMBL4698581

COC(=O)c1ncccc1-c1ccc(CN2CC(C)N[C@@H](C)C2)cc1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MLNR O43193 20/20 0.63
CYP3A4 P08684 7/20 0.61
CYP2D6 P10635 1/20 0.60
GHSR Q92847 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5131916 1.00 MLNR (0.63) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4698080 0.89 MLNR (0.63) MLNRCYP3A4CYP2D6GHSR
SCHEMBL5121342 0.88 MLNR (0.64) MLNRCYP3A4CYP2D6GHSR
SCHEMBL5126864 0.84 MLNR (0.65) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4698229 0.84 MLNR (0.65) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4699150 0.83 MLNR (0.55) MLNRCYP3A4CYP2D6GHSR
SCHEMBL5128343 0.83 MLNR (0.55) MLNRCYP3A4CYP2D6GHSR
SCHEMBL5123512 0.81 MLNR (0.46) MLNRCYP3A4CYP2D6GHSR
SCHEMBL4699108 0.78 MLNR (0.86) MLNRCYP3A4CYP2D6GHSR
SCHEMBL5130928 0.77 MLNR (0.49) MLNRCYP3A4CYP2D6GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902022-A1 PIPERAZINE HETEROARYL DERIVATES AS GPR38 AGONISTS GLAXO GROUP LIMITED (GB) 2008-03-26 EP disclosed
WO-2007007018-A1 PIPERAZINE HETEROARYL DERIVATES AS GPR38 AGONISTS GLAXO GROUP LIMITED (GB) 2007-01-18 WO disclosed