SCHEMBL470023

SCHEMBL470023

Cc1cc(-c2cnc3c(NCC4CCS(=O)(=O)CC4)cc(Oc4cccnc4)nn23)ccc1C(N)=O

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TTK P33981 16/20 0.68
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PIM1 P11309 2/20 0.42
KCNH2 Q12809 1/20 0.42
FYN P06241 1/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457795 0.92 TTK (0.81) TTKCYP3A4CYP2C9CYP2C19
SCHEMBL470040 0.91 TTK (0.69) TTKCYP3A4CYP2C9CYP2C19PIM1
SCHEMBL470035 0.90 TTK (0.55) TTKPIM1KCNH2
SCHEMBL10279709 0.89 TTK (0.54) TTKPIM1KCNH2
SCHEMBL10279711 0.89 TTK (0.60) TTKPIM1KCNH2
SCHEMBL457796 0.86 TTK (0.81) TTKCYP3A4CYP2C9CYP2C19
SCHEMBL470037 0.86 TTK (0.61) TTKPIM1KCNH2
SCHEMBL15556070 0.84 TTK (0.82) TTKCYP3A4CYP2C9CYP2C19
SCHEMBL457024 0.83 TTK (0.83) TTKCYP3A4CYP2C9CYP2C19
SCHEMBL10279263 0.83 TTK (0.51) TTKPIM1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed