SCHEMBL4701869

SCHEMBL4701869

CC([N])c1ccccc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4165369 1.00
SCHEMBL4166272 1.00
SCHEMBL27686008 0.75
Isopropylbenzene SCHEMBL27920380 0.75 TSHR (0.46)
Isopropylbenzene SCHEMBL87809 0.73 TAAR1 (0.50)
SCHEMBL908216 0.73 TAAR1 (0.50)
Isopropylbenzene SCHEMBL6568 0.73
SCHEMBL7499823 0.73 TAAR1 (0.50)
SCHEMBL169730 0.73 TAAR1 (0.50)
Isopropylbenzene SCHEMBL8431863 0.73 TAAR1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130352-A Method for producing (+) (2S,3S)-3-(2-aminophenylthio)-2-hydroxy-3(4'-methoxyphenyl)-propionic acid COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2000-10-10 US claimed
EP-0374647-B1 Process for the preparation of optically active alpha-amino-acetals BASF AG (DE) 1994-06-15 EP claimed
US-20150065738-A1 PHOSPHOROUS COMPOUND AND TRANSITION METAL COMPLEX THEREOF TAKASAGO INTERNATIONAL CORPORATION (JP) 2015-03-05 US disclosed
EP-2842959-A1 Phosphorous compound and transition metal complex thereof Takasago International Corporation (JP) 2015-03-04 EP disclosed
EP-1979308-A1 OPTICAL ISOMERS OF DIHYDRO-2,3-BENZODIAZEPINES AND THEIR STEREOSELECTIVE SYNTHESIS EGIS Gyógyszergyár Nyrt (HU) 2008-10-15 EP disclosed
US-20080036373-A1 Platinum complex and light-emitting device TAKASAGO INTERNATIONAL CORPORATION 2008-02-14 US disclosed
WO-2007077469-A1 OPTICAL ISOMERS OF DIHYDRO-2,3-BENZODIAZEPINES AND THEIR STEREOSELECTIVE SYNTHESIS EGIS GYÓGYSZERGYÁR (HU) 2007-07-12 WO disclosed
US-20060202197-A1 Platinum complex and light-emitting device TAKASAGO INTERNATIONAL CORPORATION 2006-09-14 US disclosed
CN-1062555-C Substituted benzyloxy carbonyl guanidine, its prepn. method, and application of the same as medicament and medicament containing the same HOECHST AG (DE) 2001-02-28 CN disclosed
US-6130352-A Method for producing (+) (2S,3S)-3-(2-aminophenylthio)-2-hydroxy-3(4'-methoxyphenyl)-propionic acid COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2000-10-10 US disclosed
EP-0748795-B1 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AG (DE) 2000-08-23 EP disclosed
WO-1991013865-A1 ANTIARRHYTHMIC AGENTS ISIS INNOVATION LIMITED (GB) 1991-09-19 WO disclosed
EP-0425976-A2 Cycloalkylidene dye-stuffs BASF Aktiengesellschaft (DE) 1991-05-08 EP disclosed
EP-0374647-A2 Process for the preparation of optically active alpha-amino-acetals BASF Aktiengesellschaft (DE) 1990-06-27 EP disclosed
EP-0196005-B1 PYRIDAZINONES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1989-12-20 EP disclosed
EP-0196005-A1 Pyridazinones, their preparation and pharmaceutical compositions containing them Dr. Karl Thomae GmbH (DE) 1986-10-01 EP disclosed
EP-0058341-B1 AZEPINE DERIVATIVES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1985-05-15 EP disclosed
US-4414225-A Azepine derivatives and their anti-thrombotic compositions and methods DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-11-08 US disclosed
EP-0058341-A1 Azepine derivatives, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-08-25 EP disclosed
US-4321063-A Motor fuel PHILLIPS PETROLEUM COMPANY (US) 1982-03-23 US disclosed