SCHEMBL470242

SCHEMBL470242

COc1ccccc1-c1noc(C)c1C(=O)N1CCN(c2cc(NC(=O)c3ccc(N(C)C)cc3)c(N=O)cc2C#N)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.49
MAPK1 P28482 1/20 0.49
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46
LMNA P02545 5/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
GHSR Q92847 1/20 0.42
GPBAR1 Q8TDU6 1/20 0.40
HTT P42858 1/20 0.39
MAPT P10636 1/20 0.39
TP53 P04637 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12457252 0.89 TSHR (0.48) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL470180 0.89 TSHR (0.48) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL457012 0.83 TSHR (0.56) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL470385 0.83 TSHR (0.54) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL12273682 0.83 TSHR (0.54) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL458542 0.83 TSHR (0.57) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL12523338 0.83 TSHR (0.57) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL458697 0.82 TSHR (0.55) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL456714 0.82 TSHR (0.56) TSHRMAPK1ALDH1A1KDM4EGAA
SCHEMBL10087686 0.82 TSHR (0.56) TSHRMAPK1ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033736-A1 NOVEL PIPERAZINE ANALOGS AS BROAD-SPECTRUM INFLUENZA ANTIVIRALS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-15 WO disclosed