SCHEMBL470339

SCHEMBL470339

CCNC(=O)c1ccc(-c2cnc3c(NCCN4CCOCC4)cc(Br)nn23)cc1C

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TTK P33981 13/20 0.49
PIK3CA P42336 1/20 0.43
MTOR P42345 1/20 0.43
FYN P06241 2/20 0.41
CYP3A4 P08684 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459405 0.92 TTK (0.50) TTKFYNCYP3A4
SCHEMBL10279112 0.90 TTK (0.61) TTKCYP3A4
SCHEMBL470065 0.90 TTK (0.49) TTKFYN
SCHEMBL10279532 0.86 TTK (0.55) TTKCYP3A4KDM4EMEN1ALDH1A1
SCHEMBL15555419 0.85 TTK (0.54) TTKCYP3A4KDM4EMEN1ALDH1A1
SCHEMBL10279719 0.85 TTK (0.53) TTKPIK3CAMTORCYP3A4
SCHEMBL17416374 0.85 TTK (0.65) TTKCYP3A4
SCHEMBL17416386 0.84 TTK (0.47) TTKFYN
SCHEMBL10279721 0.84 TTK (0.57) TTKFYNCYP3A4
SCHEMBL10279277 0.84 TTK (0.55) TTKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9255100-B2 Substituted imidazopyridazines BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-02-09 US disclosed
EP-2614063-B1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-01-13 EP disclosed
EP-2614063-B1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-01-13 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed