SCHEMBL4707898

SCHEMBL4707898

CC(C)c1nnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2ccccc2)n1Cc1ccccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 1/20 0.36
SLC16A1 P53985 1/20 0.36
MCTS1 Q9ULC4 1/20 0.36
PTGER4 P35408 2/20 0.36
CNR2 P34972 1/20 0.36
GRM2 Q14416 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90B1 P14625 1/20 0.36
TRAP1 Q12931 1/20 0.36
CDC7 O00311 4/20 0.35
MAP4K4 O95819 3/20 0.35
PIM1 P11309 3/20 0.35
PRKACA P17612 3/20 0.35
CDK2 P24941 3/20 0.35
GSK3B P49841 3/20 0.35
HIPK2 Q9H2X6 3/20 0.35
DAPK3 O43293 2/20 0.35
ROCK2 O75116 2/20 0.35
PRKD3 O94806 2/20 0.35
FLT3 P36888 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707214 0.89 CDC7 (0.39) SLC16A3SLC16A1MCTS1CNR2GRM2
SCHEMBL4705832 0.88 GRM2 (0.38) SLC16A3SLC16A1MCTS1CNR2GRM2
SCHEMBL4707480 0.85 GRM2 (0.38) SLC16A3SLC16A1MCTS1CNR2GRM2
SCHEMBL4707206 0.85 TACR1 (0.37) SLC16A3SLC16A1MCTS1CNR2GRM2
SCHEMBL4708151 0.85 SLC16A3 (0.36) SLC16A3SLC16A1MCTS1PTGER4CNR2
SCHEMBL4708164 0.84 IDO1 (0.36) SLC16A3SLC16A1MCTS1CNR2GRM2
SCHEMBL4707417 0.84 GRM2 (0.37) SLC16A3SLC16A1MCTS1CNR2GRM2
SCHEMBL4709645 0.83 CDC7 (0.38) SLC16A3SLC16A1MCTS1PTGER4GRM2
SCHEMBL4707454 0.83 CDC7 (0.38) SLC16A3SLC16A1MCTS1GRM2CDC7
SCHEMBL4706125 0.82 CYP19A1 (0.42) SLC16A3SLC16A1MCTS1HSP90AA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed