SCHEMBL4708166

SCHEMBL4708166

O=C(Cn1c(C(=O)N2CCOCC2)c(CN2CCC(c3c(F)cccc3Cl)CC2)c2ccccc21)OC(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
CYP2A13 Q16696 1/20 0.39
KDM4E B2RXH2 3/20 0.39
POLB P06746 2/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CNR2 P34972 3/20 0.36
CNR1 P21554 2/20 0.36
MGLL Q99685 1/20 0.36
ABHD6 Q9BV23 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
ALOX15 P16050 1/20 0.36
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4706829 0.90 KMT2A (0.41) KMT2AMEN1CYP2A13KDM4EPOLB
Trifluoroacetic Acid SCHEMBL4708162 0.89 CYP2A13 (0.41) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4706868 0.87 CYP2A13 (0.43) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4707699 0.86 KDM4E (0.43) KMT2AMEN1KDM4EPOLBTSHR
SCHEMBL4780859 0.86 KMT2A (0.44) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4779350 0.86 CYP2A13 (0.42) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4780919 0.84 CYP2A13 (0.46) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4780703 0.83 CYP2A13 (0.42) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4780706 0.82 CNR2 (0.42) KMT2AMEN1CYP2A13KDM4EPOLB
SCHEMBL4779504 0.81 KMT2A (0.40) KMT2AMEN1CYP2A13KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO disclosed
EP-1873150-A1 Fluorinated indoleamides useful as ligands of the ORL-1 receptor NIKEM RESEARCH S.R.L. (IT) 2008-01-02 EP disclosed