SCHEMBL4710149

SCHEMBL4710149

Cc1c[nH]c(-c2cc(NC(=O)c3ccc(C)c(Nc4nccc(-c5cnccn5)n4)c3)cc(C(F)(F)F)c2)n1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 16/20 0.70
BCR P11274 6/20 0.70
KDR P35968 3/20 0.70
ADORA3 P0DMS8 2/20 0.70
NR1I2 O75469 1/20 0.70
PTGS1 P23219 1/20 0.70
CHRNA4 P43681 1/20 0.70
PDE3A Q14432 1/20 0.70
KIT P10721 6/20 0.60
PDGFRA P16234 6/20 0.60
PDGFRB P09619 5/20 0.60
LYN P07948 4/20 0.60
LCK P06239 3/20 0.60
FLT3 P36888 3/20 0.60
DDR2 Q16832 3/20 0.60
LDLR P01130 2/20 0.60
PCSK9 Q8NBP7 2/20 0.60
EPHB6 O15197 1/20 0.60
CA12 O43570 1/20 0.60
CACNA1F O60840 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005305 0.91 ABL1 (0.72) ABL1BCRKDRADORA3NR1I2
Hydrochloric Acid SCHEMBL4600295 0.91 ABL1 (0.71) ABL1BCRKDRADORA3NR1I2
Hydrochloric Acid SCHEMBL1754053 0.90 ABL1 (0.70) ABL1BCRKDRADORA3NR1I2
SCHEMBL3362592 0.88 ABL1 (0.58) ABL1BCRKDRADORA3NR1I2
SCHEMBL4713847 0.86 ABL1 (0.56) ABL1BCRKDRADORA3NR1I2
Radotinib SCHEMBL3359952 0.83 ABL1 (1.00) ABL1BCRKDRADORA3NR1I2
Radotinib SCHEMBL29381661 0.83 ABL1 (1.00) ABL1BCRKDRADORA3NR1I2
Radotinib SCHEMBL29366343 0.83 ABL1 (1.00) ABL1BCRKDRADORA3NR1I2
Radotinib SCHEMBL15285797 0.82 ABL1 (0.99) ABL1BCRKDRADORA3NR1I2
Radotinib SCHEMBL30002961 0.82 ABL1 (0.99) ABL1BCRKDRADORA3NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1922309-A1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Il Yang Pharm. Co. Ltd. (KR) 2008-05-21 EP claimed
WO-2007018325-A1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF IL-YANG PHARM. CO., LTD. (KR) 2007-02-15 WO claimed
EP-1922309-A1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Il Yang Pharm. Co. Ltd. (KR) 2008-05-21 EP disclosed
WO-2007018325-A1 N-PHENYL-2-PYRIMIDINE-AMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF IL-YANG PHARM. CO., LTD. (KR) 2007-02-15 WO disclosed