SCHEMBL4710272

SCHEMBL4710272

CC1(C)CC(O)(C#N)c2cc(Br)ccc2O1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.47
CTSD P07339 2/20 0.47
AKR1B1 P15121 5/20 0.40
APP P05067 1/20 0.33
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14862455 0.80 BACE1 (0.49) BACE1CTSDAKR1B1APPTP53
SCHEMBL4711816 0.79 AKR1B1 (0.38) BACE1CTSDAKR1B1KMT2A
SCHEMBL2182582 0.79 BACE1 (0.46) BACE1CTSDAKR1B1APPMAPT
SCHEMBL4713122 0.77 AKR1B1 (0.49) BACE1CTSDAKR1B1APPSMN1; SMN2
SCHEMBL4518818 0.77 BACE1 (0.51) BACE1CTSDAKR1B1APPMAPT
SCHEMBL5333068 0.72 BACE1 (0.43) BACE1CTSDAKR1B1APPMAPT
SCHEMBL6906553 0.69 BACE1 (0.43) BACE1CTSDAKR1B1MAPTSMN1; SMN2
SCHEMBL12299613 0.68 BACE1 (0.42) BACE1CTSDAKR1B1MAPTSMN1; SMN2
SCHEMBL14053723 0.68 BACE1 (0.44) BACE1CTSDAKR1B1APP
SCHEMBL6915372 0.68 BACE1 (0.41) BACE1CTSDAKR1B1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008007210-A2 NITROGENOUS N-SUBSTITUTED 4-SPIRO-HETEROCYCLIC 2, 2 -DIMETHYLCHROMANE DERIVATIVES UNIVERSITA' DI PISA (IT) 2008-01-17 WO disclosed