SCHEMBL4712422

SCHEMBL4712422

Cc1cn(-c2ccc(C(N)=O)c(N[C@H]3CC[C@H](OC(=O)[C@H](C)NCCCN)CC3)c2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 19/20 0.67
HSP90AB1 P08238 19/20 0.67
HSP90B1 P14625 5/20 0.48
TRAP1 Q12931 5/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5148447 0.89 HSP90AA1 (0.67) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL5148446 0.89 HSP90AA1 (0.67) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL4707244 0.88 HSP90AA1 (0.68) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1745946 0.87 HSP90AA1 (0.73) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL2163746 0.87 HSP90AA1 (0.73) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1219414 0.87 HSP90AA1 (0.73) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL4709365 0.86 HSP90AA1 (0.74) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL5146989 0.86 HSP90AA1 (0.74) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1220356 0.86 HSP90AA1 (0.77) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL1220353 0.86 HSP90AA1 (0.77) HSP90AA1HSP90AB1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991525-A1 CYCLOHEXYLAMINO, BENZENE, PYRIDINE, AND PYRIDAZINE DERIVATIVES Serenex, Inc. (US) 2008-11-19 EP claimed
WO-2007101156-A1 CYCLOHEXYLAMINO, BENZENE, PYRIDINE, AND PYRIDAZINE DERIVATIVES SERENEX, INC. (US) 2007-09-07 WO claimed