SCHEMBL4713799

SCHEMBL4713799

Nc1ccccc1NC(=O)c1ccc(CCn2nc3ccc(C(F)(F)F)cc3c2N)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.55
HDAC1 Q13547 15/20 0.54
HDAC2 Q92769 5/20 0.49
ADORA2A P29274 5/20 0.47
HDAC3 O15379 3/20 0.47
ADORA1 P30542 2/20 0.47
ADORA2B P29275 1/20 0.47
HDAC10 Q969S8 1/20 0.47
BRD4 O60885 2/20 0.45
HDAC8 Q9BY41 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
NAMPT P43490 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3548819 0.91 HDAC1 (0.63) PTGS1HDAC1HDAC2
SCHEMBL3555022 0.83 HDAC1 (0.61) PTGS1HDAC1
SCHEMBL3551914 0.78 HDAC1 (0.61) PTGS1HDAC1HDAC2
SCHEMBL4761342 0.78 HDAC1 (0.51) HDAC1
SCHEMBL3548329 0.77 HDAC1 (0.63) PTGS1HDAC1HDAC2
SCHEMBL3555971 0.76 HDAC1 (0.61) PTGS1HDAC1
SCHEMBL3550053 0.76 HDAC1 (0.69) HDAC1HDAC2
SCHEMBL3551358 0.76 HDAC2 (0.59) PTGS1HDAC1HDAC2HDAC3HDAC10
SCHEMBL3557646 0.74 HDAC1 (0.61) PTGS1HDAC1HDAC2
SCHEMBL3554866 0.74 HDAC1 (0.58) PTGS1HDAC1HDAC2HDAC3HDAC10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904452-A2 HISTONE DEACETYLASE INHIBITORS Takeda San Diego, Inc. (US) 2008-04-02 EP claimed
WO-2007011626-A2 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2007-01-25 WO claimed